Ephedrine Nasal Spray & Liquid Drops Review – Where to Buy?
Ephedrine nasal sprays are common nasal decongestion treatments used to improve breathing, relieve allergy symptoms and alleviate the symptoms of sinusitis.
Ephedrine HCL nasal drops are FDA-approved for sale in the United States. But this product is subject to increased legal scrutiny due to the potential for misuse and abuse.
Use of ephedrine sprays, tablets, liquids, mists, or inhalers can help to ease a blocked or congested nose caused by a cold, rhinitis or hay fever allergies. These nose drops can be purchased without a prescription from a pharmacy, but your doctor may also prescribe them to you for treatment of a medical condition.
Ephedrine nasal drops are safe for adults and children over the age of 12 when they are used under doctor supervision. The sprays can be administered to each nostril up to 4 times per day and can be taken for up to 7 days.
While the use of this ingredient for relief or nasal congestion or lung problems is not associated with serious side effects, this product is sometimes abused or taken off-label as part of a weight loss regimen. Click here to buy ephedra supplements online legally without a prescription.
Ephedrine Nasal Sprays Review
Ephedrine HCL is commonly used as a decongestant, bronchodilator and in nasal sprays to improve breathing and reduce mucus accumulations.
Ephedrine is a stimulant ingredient that is derived from the Ephedra Sinica plant. When administered to the nose, it works by causing small blood vessels in your nasal cavity to constrict (become narrower).
This mechanism of action results in the lining of your nose becoming thinner and reduces swelling and inflammation, which can clear congestion and relieve the feeling of being blocked up.
According to one description, “Ephedrine redistributes the blood flow and causes cardiac stimulation without markedly raising the blood pressure. Sympathomimetic drugs exert their effect by vasoconstriction of the mucosal blood vessels, which in turn reduces the thickness of the nasal mucosa. However, they can give rise to a rebound phenomenon as their effects wear off, due to a secondary vasodilation with a subsequent temporary increase in nasal congestion.”
Due to the potential for side effects and adverse reactions, newer drugs and formulas are increasingly substituting ephedrine components in such products, intending to reduce potential for side effects.
Mechanism of Action
Ephedrine is defined as a sympathomimetic amine, implying that it has an influence over the sympathetic nervous system. This system in the body is responsible for functions that we can’t control such as:
- Heart rate
Ephedrine has been shown to increase stimulation of alpha and beta-adrenergic receptors in the body which can influence blood pressure, vascular constriction, and airway dilation.
It is also effective in dilating airways in the lungs, enabling easier breathing and greater intake of oxygen. Ephedrine can also influence a number of neurotransmitters in the brain including dopamine and norepinephrine (noradrenaline).
It has similar effects to adrenaline, a neurohormone that is release in the body during times of stress, excitement or danger. Like adrenaline, ephedrine HCL is a stimulant and can provide individuals using such products with bursts of energy that can last anywhere from one to six hours.
This compound is commonly taken off-label to promote fat loss, physical performance, energy enhancement and greater mental alertness. Overuse of this stimulant can cause a number of unpleasant side effects and may lead to long-term health risks.
Buy Ephedrine Nasal Drops
A number of ephedrine nasal spray products are currently available on the market, but access to these products will depend on where you live. In some countries, this ingredient is highly regulated and may not be available without a prescription.
In the United States, Canada, and the UK, you can buy ephedrine pills, liquids, sprays, mists and drops for the relief of nasal congestion However, there may be limitations to the amount you can buy at any one time over-the-counter.
For example, in the UK the Weldricks website selling the Care brand states that due t legal restrictions, a maximum of 180 mg of ephedrine can be sold in any one product.
Different formulations exist, with the most common brands providing either a 1% or 0.5% generic ephedrine HCL or sulfate solution. Drops are typically sold in a 10 mL bottle.
Ephedrine nasal drops are recommended for those dealing with the side effects and blocked nasal passages associated with colds or severe allergy symptoms.
Because of its mechanism of action, ephedrine can trigger vasoconstriction, which prompts the smaller blood vessels in the nose to constrict or narrow. In addition, it is effective in dilating mucosal lining such as those found in the lung airways as well as sinus and nasal passages.
When it comes to bronchodilator or decongestant medications, consumers may find that most ephedrine HCL formulas sold in the USA also contain a minimum of 200 mg guaifenesin.
Guaifenesin is an expectorant, used to relieve buildup of mucus in the lungs and promote drainage of mucus from the nasal passages. It is included in products to help make coughs more productive.
Dosage and Usage
Dosage and usage recommendations for ephedrine nasal spray products will differ depending on manufacturer and formulation provided. Some brands provide a 0.5% liquid solution while others provide a 1.0% solution.
According to one the directions provided with one product, “Place 1 or 2 drops into each nostril when required. Place 1 or 2 drops into each nostril when required.”
The amount you take, and frequency of dosage will depend on the condition being treated and physician instructions. Do not use more than the recommended amount of this product. Do not take more than the minimum amount required to experience desired effects.
Ephedrine can cause a stimulating effect in some users. Taking this product late in the day can make it harder to fall asleep at night.
It is suggested to discard any unused drops 2 months after opening the package and to store the product below 25°C.
Excipients in this product can include Chlorobutanol Hemihydrate, Sodium Chloride, and Purified Water. Do not use if you have an allergy or sensitivity to one of the excipients.
There is a potential for side effects with any type of medication. Use of ephedrine products is associated with a number of possible side effects, although most reports of serious adverse effects are linked to use of oral capsules and tablets, not nasal sprays.
Before taking ephedrine decongestant products, consult with a doctor to determine whether this product is safe for you. This product is contraindicated for individuals with certain medical conditions or using certain drugs and supplements.
One of the most common side effects of using ephedrine nasal drops include irritation of the nasal cavity, such as burning sensations, stinging, itching, or soreness in the nose. It can also trigger feelings of nausea and headaches.
Ephedrine can cause dizziness as well as difficulty sleeping. When taking in high dosages, this ingredient can also cause euphoria, giddiness, vomiting, sweating, muscle tremors or weakness, anxiety, restlessness, paranoid psychosis, delusions, hallucinations, excessive thirst, tachycardia, precordial pain, palpitations and difficulty in micturition.
Ephedrine may also negatively affect blood sugar levels, especially if you are diagnosed as prediabetic or diabetic and/or taking any type of diabetes medications.
This product can interact with MAOI medications and should not be given within 14 days of taking an MAOI drug. Do not use it with beta-blockers, other stimulants, Adrenergic neurone blockers, Appetite suppressants, Antipsychotics or drugs used to treat blood pressure.
Because it is unknown how ephedrine affects a developing fetus or a growing infant, such products should not be used by pregnant or breast-feeding women. This ingredient can be excreted in breast milk.
Always discuss potential risks of use with your physician, obstetrician, or pediatrician. While responsible use of ephedrine nasal sprays is generally well tolerated, this product can be misused and can cause serious side effects.
Using Ephedrine for Weight Loss
Using ephedrine nasal sprays, asthma medications or decongestant products for nonmedical purposes such as weight loss or energy enhancement can increase the risk of side effects.
The benefits of using ephedrine-based products for weight loss may not outweigh the risk of side effects in the long-term. Taking medications designed to treat nasal congestion and to promote bronchodilation for fat loss can produce unintended adverse effects due to the presence of other ingredients in many of these products.
Ephedrine acts as a Central Nervous System stimulant, causing excitation of receptors in the body that regulate metabolism, energy production, appetite control as well as mental alertness.
It has long been used to increase the rate at which your body burns fat. Research shows that it can cause your thermogenic activity to increase, meaning that you are burning more calories and converting them into heat.
This can have a modest impact on weight loss and make it easier to kick-start a diet program. However, there is a high risk of side effects when taking ephedrine in dosages that are sufficient to cause weight loss. Potential symptoms of overuse can include:
- Heart palpitations
- Difficulty urinating
- Allergic reaction
- Irregular heart rate (arrhythmia)
In extreme cases, ephedrine fat burners and diet pills have been linked to heart attacks, fatalities, strokes, seizures and other dangerous outcomes. There are safer alternatives that you can use instead.
Where to Find Ephedrine for Sale
Consumers can find a number of ephedrine nasal spray products sold through pharmacies and retail distributors in the US, and in other geographical locations around the world.
Such products are not typically available online from auction sites such as eBay and Amazon. You will also not find these products in certain states in the USA due to legal restrictions.
While usually sold over-the-counter without requiring a doctor’s prescription, in some locations you may need a prescription to legally buy this product.
Note that some bronchodilator and asthma medications that previously contained Ephedrine HCL as their active ingredient have been reformulated to remove this ingredient due to risk of side effects.
For example, many consumers mistakenly believe that the Ephrine Nasal Drops brand contains ephedrine, but this product states that Phenylephrine HCl is the active ingredient on its package. This product is sold in the USA at Walgreens and is part of their in-store Well brand.
Before you buy any preparation or brand of oral or nasal decongestant containing ephedrine spray, consult with a doctor about the potential side effects and safety warnings regarding this product.